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Tizanidine
Tizanidine

0.76
This therapeutic option reduces skeletal muscle spasticity to help with movement comfort.
Ingredient
Tizanidine
Category
Pain & Anti-Inflammatories
Availability
In Stock
Delivery Time
Airmail (14-21 days) | Trackable (5-9 days)
Shipped in a discreet, unmarked envelope with all required documents enclosed.

Product Sheet

Active Ingredient(s)
Tizanidine
Reference Brand
Zanaflex
Product Origin
Generic Product
Reference Manufacturer
Novartis
Product Form
Tablet, Capsule
Regulatory Classification
Rx
Primary Category
Pain Management
Product Category
Skeletal Muscle Relaxant
Pharmacological Class
Alpha-2 Adrenergic Agonist
Clinical Indications
Spasticity, Muscle spasm
Manufacturer Description
Formulated for muscle spasticity to manage stiffness and support physical mobility.
Mechanism of Action
Tizanidine acts as an agonist at central alpha-2 adrenergic receptors. This action increases presynaptic inhibition of motor neurons, reducing the release of excitatory amino acids and alleviating muscle spasticity.
Route of Administration
Oral
Onset Time
1–2 hours
Duration
3–6 hours
Contraindications
Concurrent use of ciprofloxacin, Concurrent use of fluvoxamine, Severe hepatic impairment, Hypersensitivity to tizanidine
Severe Adverse Events
Hepatotoxicity, Hallucinations, Severe hypotension — requires immediate medical attention
Common Side Effects
Dry mouth, Somnolence, Dizziness
Uncommon Side Effects
Hypotension, Fatigue, Bradycardia
Drug Interactions
Alcohol, Ciprofloxacin, Fluvoxamine, Oral Contraceptives, Amiodarone
Pregnancy Safety Warnings
FDA Category C: Use only if clearly needed. Breastfeeding: Not recommended.
Age Restrictions
Safety and efficacy in pediatric patients have not been established.
Storage Guidelines
Store at room temperature.
Related Products
Sirdalud, Baclofen, Flexeril
Information related to Tizanidine is compiled and periodically reviewed with reference to established medical sources and prescribing guidance. Content is provided for general reference and should be confirmed with a registered healthcare professional before use.
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