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Rapamycin
Rapamycin

3.96
It helps regulate immune responses to address key inflammatory conditions and overactivity.
Ingredient
Sirolimus
Category
Autoimmune Support
Availability
In Stock
Delivery Time
Airmail (14-21 days) | Trackable (5-9 days)
Shipped in a discreet, unmarked envelope with all required documents enclosed.

Product Sheet

Active Ingredient(s)
Sirolimus
Reference Brand
Rapamune
Product Origin
Generic Product
Reference Manufacturer
Pfizer
Product Form
Tablet, Oral Solution
Regulatory Classification
Rx
Primary Category
Autoimmune Support
Product Category
mTOR Inhibitor
Pharmacological Class
Immunosuppressant
Manufacturer Description
Formulated for organ transplant rejection prophylaxis to target immune cell activity and support graft survival.
Mechanism of Action
Sirolimus binds to the intracellular protein FKBP-12. The resulting complex inhibits the mTOR kinase, which is required for T-lymphocyte activation and proliferation in response to cytokines like IL-2.
Route of Administration
Oral
Onset Time
1–3 days
Duration
60 hours (half-life)
Contraindications
Hypersensitivity to sirolimus, Recent lung transplant
Severe Adverse Events
Nephrotoxicity, Lymphoma, Serious infections — requires immediate medical attention
Common Side Effects
Nausea, Headache, Stomatitis
Uncommon Side Effects
Hypertension, Hyperlipidemia, Anemia
Drug Interactions
Grapefruit, Cyclosporine, Ketoconazole, Rifampin, Alcohol
Pregnancy Safety Warnings
FDA Category C: Benefit must justify risk. Breastfeeding: Excretion in milk is unknown; not recommended.
Age Restrictions
Safety and efficacy established in pediatric patients 13 years and older.
Storage Guidelines
Store in the refrigerator (2°C to 8°C); tablets may be kept at room temperature.
Related Products
Rapamune, Afinitor, Zortress
Information related to Rapamycin is compiled and periodically reviewed with reference to established medical sources and prescribing guidance. Content is provided for general reference and should be confirmed with a registered healthcare professional before use.
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