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Eptus
Eptus

3.8
This key compound works to block excess hormone signaling that impacts blood vessel relaxation.
Ingredient
Eplerenone
Category
Heart & Blood Pressure
Availability
In Stock
Delivery Time
Airmail (14-21 days) | Trackable (5-9 days)
Shipped in a discreet, unmarked envelope with all required documents enclosed.

Product Sheet

Active Ingredient(s)
Eplerenone
Product Origin
Generic Brand
Product Manufacturer
Glenmark Pharmaceuticals
Product Form
Tablet
Regulatory Classification
Rx
Primary Category
Heart & Blood Pressure
Product Category
Aldosterone Receptor Antagonist
Pharmacological Class
Potassium-Sparing Diuretic
Manufacturer Description
Intended for congestive heart failure to manage fluid balance and support cardiac survival post-infarction.
Mechanism of Action
Eplerenone selectively binds to the mineralocorticoid receptor, blocking the binding of aldosterone. This prevents sodium retention and subsequent fluid accumulation, while also mitigating myocardial fibrosis and vascular damage.
Route of Administration
Oral
Onset Time
1–2 weeks
Duration
4–6 hours (half-life)
Contraindications
Hyperkalemia, Severe renal impairment, Concurrent use of strong CYP3A inhibitors
Severe Adverse Events
Renal failure, Severe hyperkalemia, Angioedema — requires immediate medical attention
Common Side Effects
Dizziness, Fatigue, Headache
Uncommon Side Effects
Hyperkalemia, Diarrhea, Abdominal pain
Drug Interactions
Alcohol, Lithium, NSAIDs, Potassium Supplements, Ketoconazole
Pregnancy Safety Warnings
FDA Category B: No evidence of fetal risk. Breastfeeding: Not known if excreted in milk.
Age Restrictions
Safety and efficacy in pediatric patients have not been established.
Storage Guidelines
Store below 25°C away from moisture.
Related Products
Inspra, Aldactone
Information related to Eptus is compiled and periodically reviewed with reference to established medical sources and prescribing guidance. Content is provided for general reference and should be confirmed with a registered healthcare professional before use.
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